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主营:防癌抗癌特殊化学品试剂
℡ 4000-520-616
℡ 4000-520-616
LKT/LEU-ENKEPHALIN/E5240/25 mg
产品编号:E5240-25mg
市  场 价:¥1500.00
场      地:美国(厂家直采)
产品分类: 其它>其它试剂>临床研究>
联系QQ:1570468124
电话号码:4000-520-616
邮      箱: info@ebiomall.com
美  元  价:$75.00
品      牌: LKT Labs
公      司:LKT Laboratories, Inc
公司分类:
LKT/LEU-ENKEPHALIN/E5240/25 mg
商品介绍
  • Description
  • ProductInfo
  • ShippingandStorage
  • Downloads
  • References

Description

Leu-enkephalinisanendogenousopioidpeptidethatactsasanagoNISTatμ-opioidreceptors(μORs)andδ-opioidreceptors(δORs).Met-enkephalinexhibitsneuromodulatory,antinociceptive/analgesic,andgastrointestinalmotilitymodulatingactivities.Likeotherendogenousopioids,leu-enkephalinmodulatesexpressionofopioidreceptorsandplaysaroleinreward/reinforcementsignaling.Leu-enkephalinincreasespainthresholdsinvivoandinhibitsgastrointestinalmusclecontractilityinotheranimalmodels,inhibitingmotilityandgastricemptying.

ProductInfo

CasNo.

58822-25-6

Purity

≥95%

Formula

C28H37N5O7

FormulaWt.

555.62

IUPACName

2-[[2-[[2-[[2-[[2-amino-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoicacid

Synonym

1-5-b-Neoendorphin(human)(9CI)

Appearance

Whitetooffwhitepowder

ShippingandStorage

StoreTemp

-20°C

ShipTemp

Ambient

Downloads

MSDS

E5240MSDSPDF

InfoSheet

E5240InfoSheetPDF

References

PopovM,AbuHammadI,BacharT,etal.Deliveryofanalgesicpeptidestothebrainbynano-sizedbolaamphiphilicvesiclesmadeofmonolayermembranes.EurJPharmBiopharm.2013Nov;85(3PtA):381-9.PMID:23791683.

CraytonR,SollerW,MattiassonA,etal.Exogenouslyadministeredopioidscontractthefemaleratintrinsicurethralsphincterinvivo.NeurourolUrodyn.2010Jun;29(5):777-82.PMID:19899147.

HolzerP.Opioidreceptorsinthegastrointestinaltract.RegulPept.2009Jun5;155(1-3):11-7.PMID:19345246.

DelBorgoMP,BlanchfieldJT,TothI.Internalisationofthemu-opioidreceptorbyendomorphin-1andleu-enkephalinisdependantonaromaticaminoacidresidues.BioorgMedChem.2008Apr15;16(8):4341-6.PMID:18329886.

品牌介绍

LKT Labs


LKT实验室是一家专注于小分子的合成、纯化和分离的生化供应公司,用于研究应用。它的产品系列展示了已知的生物活性,在广泛的研究领域,特别是癌症和神经科学中得到了广泛的应用。这些产品包括蛋白激酶抑制剂、离子通道调节剂和激活剂。


LKT Laboratories is a biochemical supply company focused on the synthesis, purification, and isolation of small molecules for research applications. Its range of products exhibit known biological activities that have found uses in a wide array of research fields, especially cancer and neuroscience. These products include protein kinase inhibitors, ion channel modulators, and activators.


品牌

货号

名称

规格

LKT Labs

444912-48-5

(2-iodo-5-nitrophenyl)-[1-[(1-methylpiperidin-2-yl)methyl]indol-3-yl]methanone

1mg 5mg 25mg

LKT Labs

 294646-77-8

(R)-CR8

1mg 5mg

LKT Labs

2377-31-3

(Z)-1,-BIS(2-METHOXY-5-(TRIFLUOROMETHYL)PHENYL)DIAZENE OXIDE

1mg 5mg 25mg

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